阻害剤について


※上記の広告は60日以上更新のないWIKIに表示されています。更新することで広告が下部へ移動します。

NMDAR

  AP-5------NMDAR antagonist

  MK-801--NMDAR blocker (開口チャンネル阻害)

  CPP------NMDAR antagonist

  Ifenprodil (3μM) NR2B-containing receptor

 

AMPAR

  NBQX----AMPAR inhibitor

 

AMPAR+Kainate receptor

  CNQX and DNQX

 

CaM

  W7

  Calmidazolium

 

CaMkII

  KN62

  KN93 (0.5μM)

 

mGluR

 DHPG  mGluR selective angonist

 MCPG mGluR antagonist

 MPEP mGluR antagonist

 

L-type channel blocker

  Nimodipine

  Nifedipine

 

GABA receptor

  picrotoxin (PCTX) GABAa receptor antagonist

  Gabazine GABAa receptor blocker

 

Dopamine receptor

  PD168077--- dopamine agonist, especially D4 receptor

  L745870 -----dopamine receptor antagonist, especially D4 receptor

 

Voltage-gated sodium  channel antagonist

  TTX (0.5μM)---action potential blocker

 

Other

Anisomycin: protein synthesis inhibitor

Calyculin A:phosphatase inhibitor

U0126:MEK inhibitor

Cholesterol inhibitor:U18666A ---cholesterol transport

V型ATPase:Bafilomycin

Actin:

latrunculin A--- inhibitor of actin reorganization: This binds within the cleft of actin monomer near ATP binding site.

cytochalasinD-N-terminal region binging: inhibitor for elongation and polymerization of actin

K252a PI(3,4)P2 inhibitor SHIP2 inihibitor